首页> 外国专利> COMPOSITION COMPRISING (±)-5-ETHYLDIHYDRO-5-(1-METHYLBUTYL)-2-THIOXO 4,6(1H,5H)-PYRIMIDINEDIONE DISSOLVED IN 2,5-DI-O-METHYL-1,4:3,6-DIANHYDRO-D-GLUCITOL

COMPOSITION COMPRISING (±)-5-ETHYLDIHYDRO-5-(1-METHYLBUTYL)-2-THIOXO 4,6(1H,5H)-PYRIMIDINEDIONE DISSOLVED IN 2,5-DI-O-METHYL-1,4:3,6-DIANHYDRO-D-GLUCITOL

机译:包含(±)-5-乙基二氢-5-(1-甲基丁基)-2-硫代氧杂分解成2,5-二-O-甲基-1,4:3,6的4,6(1H,5H)-嘧啶二酮的组合物-二氨基D-葡糖醇

摘要

This invention relates to an injectable ready-to-use formulation of THIOPENTAL the chemical name of which is (±)-5-Ethyldihydro-5-(1-methylbutyl)-2-thioxo 4,6(1H,5H)-Pyrimidinedione and which is used in inducing anaesthesia. The invention utilizes crysalline THIOPENTAL which is dissolved in 2,5-di-O-methyl-1,4:3,6-dianhydro-D-glucitol, which is a biologically acceptable non-toxic solvent, for administration parenterally to mammals including humans.
机译:本发明涉及THIOPENTAL的可注射即用制剂,其化学名称为(±)-5-乙基二氢-5-(1-甲基丁基)-2-硫代4,6(1H,5H)-嘧啶二酮和用于诱导麻醉。本发明利用了溶解在2,5-二-O-甲基-1,4:3,6-二脱水-D-葡萄糖醇中的晶状体THIOPENTAL,其是生物学可接受的无毒溶剂,用于胃肠道外给药给包括人在内的哺乳动物。

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