首页> 外国专利> PHARMACEUTICAL COMPOSITION FOR TREATMENT OF LIVER CANCER CONTAINING DIAMINEDITHIOL-RADIOACTIVE RHENIUM COMPLEX AND LIPIODOL, PRODUCTION AND KIT FOR PRODUCTION THEREOF

PHARMACEUTICAL COMPOSITION FOR TREATMENT OF LIVER CANCER CONTAINING DIAMINEDITHIOL-RADIOACTIVE RHENIUM COMPLEX AND LIPIODOL, PRODUCTION AND KIT FOR PRODUCTION THEREOF

机译:用于治疗含双氨基二巯基-放射性AC配合物和利多多的肝癌的药物组合物,生产及其生产用试剂盒

摘要

PURPOSE: A composition for the treatment of liver cancer containing diaminedithiol-radioactive and a kit for producing the same are provided. Therefore, the composition exhibits excellent effect on treating liver cancer without side effects when injected to liver cancer patients through the hepatic artery. CONSTITUTION: Diaminedithiol, a reducing agent and an auxiliary agent are reacted with radioactive rhenium to produce a radioactive rhenium complex, which is dissolved in lipiodol to produce the titled composition represented by formula 1, wherein the reducing agent and auxiliary agent are tin chloride and tartaric acid respectively. In formula, R1 to R12 are each independently H or C1-5 lower alkyl.
机译:目的:提供一种包含二胺二硫醇放射性的治疗肝癌的组合物及其制备试剂盒。因此,当通过肝动脉注射给肝癌患者时,该组合物表现出优异的治疗肝癌的效果而没有副作用。组成:二胺二硫醇,还原剂和助剂与放射性rh反应生成放射性rh络合物,将其溶解在碘油中制得式1所示的标题组合物,其中还原剂和助剂为氯化锡和酒石酸分别酸。式中,R 1〜R 12分别独立地为H或C 1-5的低级烷基。

著录项

  • 公开/公告号KR20010053908A

    专利类型

  • 公开/公告日2001-07-02

    原文格式PDF

  • 申请/专利权人 SEOUL NATIONAL UNIVERSITY HOSPITAL;

    申请/专利号KR19990054469

  • 发明设计人 JUNG JAE MIN;

    申请日1999-12-02

  • 分类号A61K33/24;

  • 国家 KR

  • 入库时间 2022-08-22 01:13:26

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