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Tricyclic pyrazolo-pyridazinone analogues as GAGA-A receptor ligands
Tricyclic pyrazolo-pyridazinone analogues as GAGA-A receptor ligands
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机译:三环吡唑并哒嗪酮类似物作为GAGA-A受体配体
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摘要
Pyrazolo[4,3-c]pyridazin-3-one analogues, represented byare selective ligands for GABAA receptors, in particular having high affinity for the alpha2 and/or alpha3 subunit thereof, are useful in the treatment of anxiety and convulsions.
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