首页> 外国专利> Modified release formulations containing (R)-1-(10,11-dihydro-5H-Dibenzoamp;lsqb;a,damp;rsqb;cyclohepten-5-ylidene)-1propyl)-3-piperidinecarboxylic acid

Modified release formulations containing (R)-1-(10,11-dihydro-5H-Dibenzoamp;lsqb;a,damp;rsqb;cyclohepten-5-ylidene)-1propyl)-3-piperidinecarboxylic acid

机译:含有(R)-1-(10,11-二氢-5H-二苯并(a,d]环庚-5-亚烷基)-1丙基)-3-哌啶羧酸的调释制剂

摘要

Modified release formulations with zero-order drug release containing (R)-1-(3-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-ylidene)-1-propyl)-3-piperidinecarboxylic acid, or a pharmaceutically acceptable salt thereof, dispersed in a polymeric matrix having at least one release rate controlling polymer are useful in treating disorders related to both neurogenic inflammation and non-insulin-dependent diabetes mellitus (NIDDM).
机译:含有(R)-1-(3-(10,11-Dihydro-5H-dibenzo[ a,d]环庚-5-亚烷基)-1-丙基)-3-哌啶羧酸的零级药物释放的调释制剂分散在具有至少一种控制释放速率的聚合物的聚合物基质中的或其药学上可接受的盐可用于治疗与神经源性炎症和非胰岛素依赖型糖尿病(NIDDM)相关的疾病。

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