1-(3-BENZYLOXYPROPYL)-5-(2-SUBSTITUTED PROPYL) INDOLINE DERIVATIVE AND METHOD FOR USING THE SAME

摘要

PROBLEM TO BE SOLVED: To provide a new 1-(3-benzyloxypropyl)-5-(2-substituted propyl)indoline derivative useful as a production raw material for pharmaceuticals and provide a method for the use of the derivative.;SOLUTION: The 1-(3-benzyloxypropyl)-5-(2-substituted propyl) indoline derivative is expressed by formula (I) (R is carboxy, carbamoyl, amino or a group of formula (II); and the carbon atom labeled with *1 has R configuration or RS configuration provided that R is carboxy when the carbon atom labeled with *1 has RS configuration). The invention further provides a method for the production of an indoline derivative expressed by formula (A) and useful as an agent for the treatment of dysurea by using the compound of formula (I).;COPYRIGHT: (C)2002,JPO