首页> 外国专利> Salt of a compound of piridopirazina or a solvate thereof, The Salt Crystals, a process for producing such crystalsThe composicionesterapeuticas containing such a compound and the use thereof for the preparation of Drugs and therapeutic compositions

Salt of a compound of piridopirazina or a solvate thereof, The Salt Crystals, a process for producing such crystalsThe composicionesterapeuticas containing such a compound and the use thereof for the preparation of Drugs and therapeutic compositions

机译:吡吡吡嗪酮化合物的盐或其溶剂化物,盐晶体,制备此类晶体的方法,包含此类化合物的组合酯类药剂及其在制备药物和治疗组合物中的用途

摘要

Describes a piridopirazina Salt of a Compound, which has the following formula (1) and its Crystal, which are very successful in terms lasolubilidad and stability.More particularly, it provides the compound of the above formula, its solvate and its crystals.It also describes lapreparacion Said Compounds, the use thereof for preparing Drugs and therapeutic compositions containing such compounds.(1) the compounds possess Inhibitory activity of fosfodiestearasa IV, the production of tumor necrosis factor Production, the production of interferons and interleukins,So that they are useful for treating various diseases such as hepatitis and trachoma.
机译:描述了具有以下式(1)的化合物的吡吡并吡嗪酸盐及其晶体,它们在拉索比利德和稳定性方面非常成功,更具体地说,它提供了上式的化合物,其溶剂化物及其晶体。描述了制备上述化合物,其在制备药物中的用途以及包含此类化合物的治疗组合物。(1)该化合物具有fosfodiestearasa IV的抑制活性,肿瘤坏死因子的产生,干扰素和白介素的产生,因此它们是有用的用于治疗各种疾病,例如肝炎和沙眼。

著录项

  • 公开/公告号AR020668A1

    专利类型

  • 公开/公告日2002-05-22

    原文格式PDF

  • 申请/专利权人 FUJISAWA PHARMACEUTICAL CO. LTD.;

    申请/专利号AR1999P104887

  • 发明设计人

    申请日1999-09-28

  • 分类号C07D471/04;A61K31/4985;A61K45/00;A61P1/16;A61P11/00;A61P11/06;A61P27/02;A61P27/06;A61P27/14;A61P31/18;A61P37/08;A61P43/00;

  • 国家 AR

  • 入库时间 2022-08-22 00:46:30

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