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DERIVATIVES OF BENZIMIDAZOLE STIRIL AS INHIBITORS OF PROLIFERATION OF SMALL CELLULAR CELLS
DERIVATIVES OF BENZIMIDAZOLE STIRIL AS INHIBITORS OF PROLIFERATION OF SMALL CELLULAR CELLS
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机译:苯并咪唑类衍生物作为小细胞增殖的抑制剂
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摘要
Disclosed herein are compounds of the formula:whereinR is phenyl or substituted phenyl;or R is furyl, pyridyl or quinolinyl;R1 and R2 are hydrogen, halogen, alkyl, alkoxy, nitro, carboxyl, alkoxy-carbonyl or aryloxycarbonyl;R3 is hydrogen, alkyl, aryl or arylalkyl;R4 and R5 are hydrogen or alkyl;or a pharmaceutically acceptable salt thereof, which are useful as inhibitors of smooth muscle cell proliferation.
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机译:本文公开了下式的化合物:其中R是苯基或取代的苯基;或R是呋喃基,吡啶基或喹啉基; R1和R2是氢,卤素,烷基,烷氧基,硝基,羧基,烷氧基-羰基或芳氧基羰基; R3是氢,烷基,芳基或芳基烷基; R 4和R 5为氢或烷基;或其药学上可接受的盐,其可用作平滑肌细胞增殖的抑制剂。
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