首页> 外国专利> THIOXYNDOL DERIVATIVES, PHARMACEUTICAL COMPOSITION CONTAINING SAID DERIVATIVES AND ACTIVE INGREDIENTS OF MEDICAMENTS FOR THE STIMULATION OF CONTRACEPTION AND TREATMENT OF DISFUNCTIONAL BLEEDING WITH CARCIN AND ADENOCARCIN

THIOXYNDOL DERIVATIVES, PHARMACEUTICAL COMPOSITION CONTAINING SAID DERIVATIVES AND ACTIVE INGREDIENTS OF MEDICAMENTS FOR THE STIMULATION OF CONTRACEPTION AND TREATMENT OF DISFUNCTIONAL BLEEDING WITH CARCIN AND ADENOCARCIN

机译:噻吩酚衍生物,包含所述衍生物的药物组合物和药物的活性成分,用于刺激宫缩抑素和腺上腺皮质激素的功能障碍性出血的避孕和治疗

摘要

This invention relates to compounds which are agonists of the progesterone receptor which have general structures (1) or (2) wherein the substituents are as defined; or a pharmaceutically acceptable salt thereof, as well as methods of using these, compounds to induce contraception or treat progesterone-related carcinomas and adenocarcinomas. , (1) , (2)
机译:本发明涉及作为孕酮受体激动剂的化合物,其具有通式(1)或(2)的结构,其中取代基如上所定义;或其药学上可接受的盐,以及使用这些化合物的方法,以诱导避孕或治疗与孕激素有关的癌和腺癌。 ,(1),(2)

著录项

  • 公开/公告号UA73499C2

    专利类型

  • 公开/公告日2002-03-15

    原文格式PDF

  • 申请/专利权人 LIGAND PHARMACEUTICALS INC.;WYETH;

    申请/专利号UA20010117770

  • 发明设计人

    申请日2000-05-01

  • 分类号C07D209/08;A61K31/404;A61P5/36;C07D209/30;C07D209/40;

  • 国家 UA

  • 入库时间 2022-08-22 00:43:29

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