INTRAMOLECULAR GLYCOSIDATION PROCESS FOR THE SYNTHESIS OF (2R, 2-ALPHA-R, 3A)-2-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY-3-(4-FLUOROPHENYL)-1,4-OXAZINE

摘要

The present invention is concerned with novel processes for the preparation of (2R-cis)-2-[[1-[3.5-bis(trifluoromethyl)phenyl]ethenyl]oxy]-3-(4-fluorophenyl)-4-(phenylmethyl)mopholine. This compound is useful as an intermediate in the synthesis of compounds which possess pharmacological activity.