首页> 外国专利> USE OF 11- (3-DIMETHYLAMINOPROPYLIDES) -6.11-DIHYDRODIBENCE B, E OXEPIN-2-ACETIC ACID AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS FOR THE PRODUCTION OF A MEDICINE FOR THE TREATMENT, NEDULATION, NEDULATION, NEDULATION, NEDULATION, NEDERATION, NEDULATION, NEDICULATION, NEDERATION, NON-DENTALIZATION

USE OF 11- (3-DIMETHYLAMINOPROPYLIDES) -6.11-DIHYDRODIBENCE B, E OXEPIN-2-ACETIC ACID AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS FOR THE PRODUCTION OF A MEDICINE FOR THE TREATMENT, NEDULATION, NEDULATION, NEDULATION, NEDULATION, NEDERATION, NEDULATION, NEDICULATION, NEDERATION, NON-DENTALIZATION

机译:使用11-(3-二甲基氨基丙酸酯)-6.11-二氢[B,E]氧杂环丁-2-乙酸及其药学上可接受的盐来生产用于治疗,消融,消融,消融,消融,结缔,结扎,结扎的药物,根除,求和,非去基化

摘要

Ophthalmic formulations containing as an active ingredient 11-(3-dimethylaminopropylidene) -6,11-dihydrodibenz[b,e]oxepin-2-acetic acid or a pharmaceutically acceptable salt thereof are useful for inhibiting cytokine release (e.g., IL-6 and IL-8) from human ocular cells. Such formulations can be used to treat or prevent ocular neovascularization and non-allergic inflammatory disorders such as dry-eye, keratitis, blepharitis, uveitis and inflammation related to infection.
机译:含有11-(3-二甲基氨基亚丙基)-6,11-二氢二苯并[b,e]氧杂环丁-2-乙酸或其药学上可接受的盐作为活性成分的眼科制剂可用于抑制细胞因子的释放(例如IL-6和IL-8)来自人眼细胞。此类制剂可用于治疗或预防眼新血管形成和非过敏性炎症性疾病,例如干眼症,角膜炎,睑缘炎,葡萄膜炎和与感染有关的炎症。

著录项

  • 公开/公告号DE69900207T2

    专利类型

  • 公开/公告日2001-11-22

    原文格式PDF

  • 申请/专利权人 ALCON LABORATORIES INC.;

    申请/专利号DE1999600207T

  • 发明设计人 YANNI M.;GAMACHE A.;WEIMER K.;

    申请日1999-06-15

  • 分类号A61K31/335;

  • 国家 DE

  • 入库时间 2022-08-22 00:24:42

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