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Preparation and drug composition of bis-benzyl-isoquinoline class alkaloids
Preparation and drug composition of bis-benzyl-isoquinoline class alkaloids
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机译:双苄基异喹啉类生物碱的制备及药物组成
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摘要
This invention relates to the preparation of bis-isoquinoline derivatives of general formula (I) and salts thereof, which possesses multi-drug resistance (MDR) reversal activities. Drug compositions and formulations comprising bis-isoquinoline derivatives of general formula (I) and salts thereof are provided for use as sensitivity enhancers in cancer chemotherapy. Methods for inhibiting MDR by treatment with bis-isoquinoline derivatives are also provided.
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