首页> 外国专利> 2- 4-(NAPHTALIN-2-YL)-THIAZOL-2-YLAMINOCARBONYL BENZOIC ACID AND 2- 4-(NAPHTALIN-2-YL)-PYRIMIDIN-2-YLAMINOCARBONYL BENZOIC ACID AND ADDITIONAL COMPOUNDS SERVING AS TELOMERASE INHIBITORS FOR USE IN TUMOR THERAPY

2- 4-(NAPHTALIN-2-YL)-THIAZOL-2-YLAMINOCARBONYL BENZOIC ACID AND 2- 4-(NAPHTALIN-2-YL)-PYRIMIDIN-2-YLAMINOCARBONYL BENZOIC ACID AND ADDITIONAL COMPOUNDS SERVING AS TELOMERASE INHIBITORS FOR USE IN TUMOR THERAPY

机译:2- 4-(萘酚-2-基)-噻唑-2-基氨基碳酰苯甲酸和2-4-萘酚(2-萘基)-嘧啶-2-基氨基苯甲酸和另外的化合物,用作端粒酶抑制剂,用于肿瘤治疗治疗

摘要

The invention relates to the use of carboxylic acid derivatives of general formula (I) R1 - A - B - R2, in which R1, R2, A and B are defined as per Claim No. 1, and to their isomers and salts, particularly their physiologically compatible salts, which have an inhibitory effect on the telomerase. The invention also relates to a method for producing said derivatives, to medicaments containing these compounds, and to their use and production thereof.
机译:本发明涉及通式(I)的羧酸衍生物的用途,其中R 1,R 2,A和B如权利要求1所定义,R 1 -A B -R 2,及其异构体和盐,特别是它们的生理相容性盐,它们对端粒酶具有抑制作用。本发明还涉及制备所述衍生物的方法,涉及包含这些化合物的药物,及其用途和生产。

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