首页> 外国专利> 3 - substituted pyrazoles Insecticides and acaricides; method for the control of Insects or mites; method for Protection of a Plant; a method for Protection of Wood, Wood Products and wooden structures; composition; and a process for the preparation of these compounds

3 - substituted pyrazoles Insecticides and acaricides; method for the control of Insects or mites; method for Protection of a Plant; a method for Protection of Wood, Wood Products and wooden structures; composition; and a process for the preparation of these compounds

机译:3-取代的吡唑类杀虫剂和杀螨剂;防治昆虫或螨虫的方法;植物保护方法;一种保护木材,木制品和木制结构的方法;组成;以及这些化合物的制备方法

摘要

3 - substituted pyrazoles of formula (1), in which the variables and the index have the following Meanings: R1 is Hydrogen, halogen, alkyl of C1 - 6 - 6, haloalquilo C1, C2 alquenilo - 6 - 6, haloalquenilo Alquiltio C1 - C2, C1 - 6, 6 - alkoxy alkyl C1 Alquiltio C1 - 4, 6 - c1-4 alkyl or Fen What is not replaced or substituted with 1 to 3 groups ra ra is Halogen, Nitro, cyano,Rent haloalquilo C1 C1 - 6, - 6, - 6 haloalquiltio Alquiltio C1, C1 - 6, 6 - alkoxy or haloalcoxi C1 C1 - 6; R2 is Hydrogen, halogen, alkyl of C1 - 6 - 6, haloalquilo C1, C2 alquenilo haloalquenilo - 6 - 6, C2 is not replaced or phenyl or substituted with 1 to 3 groups ra is Hydrogen, Hydroxy, CIANO Rhone, halogen, alkoxy, Nitro, haloalcoxi C1 C1 - 6, - 6, - 6 Alquiltio alqueniloxi C2, C1 - 6Haloalquiltio alquilsulfinilo C1 C1 - 6, - 6, - 6 aminotiocarbonilo alquilsulfonilo C1, C1, hidroxicarbonilo, alcoxicarbonilo - 6 or aminocarbonilo; b is Hydrogen, Hydroxy, amino, cyano, Nitro alkyl or Halogen; C1 - 6 unsubstituted or substituted with 1 to 3 and cyano groups selected from Halogen, alkoxy C1 - 6 unsubstituted or substituted with 1 to 3 groups selected from Halogen, cyano,Alquenilo alcoxicarbonilo C1 and C2 - 4 - 6 - alquenilo c2-4; alquenilo C2 6 unsubstituted or substituted with 1 to 3 groups selected from Halogen and cyano; alqueniloxi Alquiltio C1 - C2 - 6, 6, 6 alcoxitiocarboniltio haloalquilo C1, C1 C1 - 6 - 6, alcoxicarbonil c1-4 alkoxy, alcoxicarbonil C1 - 6 - Alquiltio c1-4, Quilsulfinilo alquilsulfonilo C1 C1 - 6 - 6, aminotiocarbonilo, nr3r4,Chor5 or n = n = chnr5; R3 and R4 are each independently Hydrogen, alkyl alcoxicarbonil C1 C1 - 6 - 6 - [(c1-4 alkyl, alcoxicarbonil C1 - 6) (alquenil C2 - 4)] c1-4 alkyl, alcoxicarbonilo C1 C2 - 4 - 6 - alquenilo, alquilcarbonilo C1 6, cicloalquilcarbonilo alquilaminocarbonilo C1 - C3 - 7, 6, 6 - Di - (alkyl C1 Aminocarbonilo), alcoxicarbonilo C1 - 6Alcoxiaminosulfonilo C1 - 6 or di - (C1 - alkoxy alkyl aminosulfonilo 6); R5 is C1 - 6 - 6, haloalquilo C1 or fenilalquilo c1-4; Q is Hydrogen, halogen, Nitro, haloalquilo alquilamino C1 C1 - 4 - 6, 6 - alkoxy dialquilamino C1, C1 C1 - 6 - 6, haloalcoxi or alqueniloxi C2 - 6; X is Hydrogen, halogen, haloalquilo C 1 - 6.Alkoxy or haloalcoxi C1 C1 - 6 - 6; and is Hydrogen, halogen, alkoxy - 6 haloalquilo C1, C1 and C1 - 6 - 6 haloalcoxi; Z is Hydrogen, halogen, alkoxy haloalquilo C1 - 6 - 6 or haloalcoxi C1, C1 - 6; n or M is Cr6; R6 is Hydrogen, Nitro, Halogen or haloalquilo c1-4; and N is 0, 1, 2, 3 or 4; under the condition of When R1 is Hydrogen,N is not Zero; method for the control of insects and mites; method for the Protection of a Plant; a method for Protection of Wood, Wood Products and wooden structures; composition; and a process for the preparation of these compounds.These compounds are also used to treat, manage, prevent and protect against infection caused by Arthropods and arachnids and endo ectoparasu00edticos.The Procedure for the preparation of compounds of formula (2), where a is B is amino and cyano compounds is that of formula (3) are reacted with malononitrile in the presence of a base, where the values of the substituents are mentioned above).
机译:式(1)的3-取代的吡唑,其中变量和指数具有以下含义:R1是氢,卤素,C1-6-6的烷基,卤代alquilo C1,C2烷基--6-6,卤代烷基Cal1- C2,C1-6,6-烷氧基烷基C1 Alquiltio C1-4,6-C1-4烷基或芬芳未被1-3个基团取代或取代的基团是卤素,硝基,氰基,Rent haalalquilo C1 C1-6 ,-6,-6卤代烷Al C1,C1-6,6-烷氧基或卤代甲氧C1 C1-6; R2是氢,卤素,C1-6-6的烷基,卤代alquilo C1,C2烷基卤代卤代烷基-6-6,C2没有被取代或未被苯基或被1-3个基团取代ra是氢,羟基,CIANO罗纳,卤素,烷氧基,硝基,卤代烷C1-6--6-6 Alquiltio alqueniloxi C2,C1-6卤代烷Alquilsulfinilo C1-6--6-6氨基噻碳基alquilsulfonilo C1,C1,hidroxicarbonilo,alcoxicarbonilo-6或氨基碳素; b是氢,羟基,氨基,氰基,硝基烷基或卤素; C1-6未取代或被1-3取代的氰基,或选自卤素,烷氧基的C1-6未取代或被1-3取代的卤素,氰基,Alquenilo alcoxicarbonilo C1和C2-4-6-alquenilo c2-4取代的烷氧基; Alquenilo C 2 6未取代或被1-3个选自卤素和氰基的基团取代; alqueniloxi Alquiltio C1-C2-6,6,6 alcoxitiocarboniltio haloalquilo C1,C1 C1-6-6,alcoxicarbil c1-4 alkoxy,alcoxicarbil C1-6-Alquiltio c1-4,Quilsulfinilo alquilsulfonilo C1 C1-6-6,6,aminotiocarbonilo4, ,Chor5或n = n = chnr5; R 3和R 4各自独立地为氢,烷基烷基锡碳环C 1-6-6-[((c1-4烷基,羟基锡碳环C1-6-(alquenil C2-4))] c1-4烷基,羟基锡碳环C 1 -C 2-4-6-羟基铝,alquilcarbonilo C1 6,cicloalquililoilo alquilaminocarbonilo C1-C3-7、6、6-Di-(烷基C1 Aminocarbonilo),alcoxicarbonilo C1-6 Alcoxiaminosulfonilo C1-6或di-(C1-烷氧基烷基氨基磺酰基6); R5是C1-6-6,卤代alquilo C1或fenilalquilo c1-4; Q为氢,卤素,硝基,卤代alquiamino C1 -C1-6-6、6-烷氧基二代氨基C1,C1-6-6-6,卤代alcoxi或alqueniloxi C2-6; X是氢,卤素,卤代喹啉C 1-6烷氧基或卤代烷氧基C1 C1-6-6;且为氢,卤素,烷氧基-6卤代alquilo C1,C1和C1-6-6卤代烷Z为氢,卤素,烷氧基卤代alquilolo C1-6-6或卤代烷氧基C1,C1-6; n或M为Cr 6; R6是氢,氮,卤素或卤代alquilo c1-4; N为0、1、2、3或4;当R1为氢时,N不为零;防治昆虫和螨虫的方法;植物保护方法;一种保护木材,木制品和木制结构的方法;组成;这些化合物还用于治疗,控制,预防和预防节肢动物,蜘蛛纲动物和内生opa虫引起的感染。式(2)化合物的制备方法如下: a是B是氨基,且氰基化合物是式(3)的氰基化合物与丙二腈在碱的存在下反应,其中取代基的值如上所述)。

著录项

  • 公开/公告号AR036631A1

    专利类型

  • 公开/公告日2004-09-22

    原文格式PDF

  • 申请/专利权人 BASF AKTIENGESELLSCHAFT;

    申请/专利号AR2002P103615

  • 发明设计人

    申请日2002-09-25

  • 分类号C07D231/12;A01N43/48;A61K31/415;A61K31/4155;C07D231/16;C07D231/18;C07D231/22;C07D231/28;C07D231/38;C07D401/04;

  • 国家 AR

  • 入库时间 2022-08-21 23:12:22

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