首页> 外国专利> Methods for treating heterozygous familial hypercholesterolemia, and for reducing ldl-c, elevating hdl-c, reducing apo b and elevating apo a-1 in a patient suffering from heterozygous familial hypercholesterolaemia, and use of (e) -7- 4 - (4-fluorophenyl) -6-isopropyl-2- methyl (methylsulfonyl) amino pyrimidin-5-yl (3r, 5s) -3,5-dihydroxyhept-6-enoic acid or a pharmaceutically acceptable salt of same

Methods for treating heterozygous familial hypercholesterolemia, and for reducing ldl-c, elevating hdl-c, reducing apo b and elevating apo a-1 in a patient suffering from heterozygous familial hypercholesterolaemia, and use of (e) -7- 4 - (4-fluorophenyl) -6-isopropyl-2- methyl (methylsulfonyl) amino pyrimidin-5-yl (3r, 5s) -3,5-dihydroxyhept-6-enoic acid or a pharmaceutically acceptable salt of same

机译:治疗杂合性家族性高胆固醇血症患者的杂合子家族性高胆固醇血症,降低ldl-c,升高hdl-c,降低apo b和升高apo a-1的方法以及(e)-7- [4-( 4-氟苯基)-6-异丙基-2- [甲基(甲基磺酰基)氨基]嘧啶-5-基](3r,5s)-3,5-二羟基庚基6-烯酸或其药学上可接受的盐

摘要

"METHODS TO TREAT HETEROZYGOTIC FAMILY HYPERCOLESTEROLEMIA, AND TO REDUCE LDL-C, RAISE HDL-C, REDUCE AFTER A-1 TO A PATIENT WHO HIGH TO FAMILY HYPERCOLESTEROLEMALIA, HETEROZYROTIC FAMILY, HYPEROZETIC FAMILY, 4- (4-FLUOROFENI) -6-ISOPROPIL-2- [METHYL (METHYLSULFONYL) AMINO] PYRIMIDIN-5-IL] (3R, 5S) -3,5-DI-HYDROXIHEPT-6-ENOIC OR OF A PHARMACEUTICALLY ACCEPTABLE SALT THE SAME". The invention provides a method for treating heterozygous familial hypercholesterolaemia by administering the compound (E) -7- [4- (4-fluorophenyl) -6-isopropyl-2- [methyl (methylsulfonyl) amino] pyrimidin-5-yl ] (3R, 5S) -3,5-dihydroxyhept-6-enoic acid or a pharmaceutically acceptable salt thereof.
机译:“治疗杂合子家族性高胆固醇血症并减少LDL-C,提高HDL-C的方法,可降低A-1患者至家族性高胆固醇血症,杂合子家族,高合子6-6-家族的患者ISOPROPIL-2- [甲基(甲基亚磺酰基)氨基] PYRIMIDIN-5-IL](3R,5S)-3,5-DI-HYDROXIHEPT-6-ENOIC或相同的药用盐。本发明提供了通过给予化合物(E)-7- [4-(4-氟苯基)-6-异丙基-2- [甲基(甲磺酰基)氨基]嘧啶丁-5-基](3R)治疗杂合性家族性高胆固醇血症的方法,5S)-3,5-二羟基庚基6-烯酸或其药学上可接受的盐。

著录项

  • 公开/公告号BR0115511A

    专利类型

  • 公开/公告日2003-12-30

    原文格式PDF

  • 申请/专利权人 ASTRAZENECA AB;

    申请/专利号BR20010115511

  • 发明设计人 ALI RAZA;HOWARD GERARD HUTCHINSON;

    申请日2001-11-16

  • 分类号A61K31/505;A61P3/06;

  • 国家 BR

  • 入库时间 2022-08-21 23:12:14

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