首页> 外国专利> NOVEL CRYSTAL FORM OF ANHYDROUS 7-(1α.5α.6α-6-AMINO-3-AZABICYCLO3.1.0HEX-3-YL)-6-FLUORO-1,(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-4-OXO-1, 8-NAPHTHYRIDINE-3-CARBOXYLIC ACID, METHANESULFONIC ACID, METHANESULFONIC ACID SALT

NOVEL CRYSTAL FORM OF ANHYDROUS 7-(1α.5α.6α-6-AMINO-3-AZABICYCLO3.1.0HEX-3-YL)-6-FLUORO-1,(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-4-OXO-1, 8-NAPHTHYRIDINE-3-CARBOXYLIC ACID, METHANESULFONIC ACID, METHANESULFONIC ACID SALT

机译:无水7-([[1α.5α.6α] -6-AMINO-3-AZABICYCLO [3.1.0] HEX-3-YL)-6-FLUORO-1,(2,4-DIFLUOPHOHENYL)-1的新晶体形式,4-二氢-4-OXO-1,8-萘啶-3-羧酸,甲磺酸,甲磺酸盐

摘要

Theanhydrate of y-9[l1a, 5a, 6a, 6--amino-3-azabicyclo[3.1.0]hex-3-yl-6-fluoro-l-(2,4-difluorophenyl)-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, methanesulfonic acid salt has advantageous stability for formulation as an antibacterial agent.
机译:y-9 [l1a,5a,6a,6--氨基-3-氮杂双环[3.1.0]己-3-基-6-氟-1-(2,4-二氟苯基)-1,4-二氢的酐-4-氧代-1,8-萘啶-3-羧酸,甲磺酸盐对于配制成抗菌剂具有有利的稳定性。

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