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Inhibitor of human myeloid leukemia on base of asymmetric cobalt trichloroacetate dimer

机译:基于不对称三氯乙酸钴二聚体的人骨髓白血病抑制剂

摘要

the invention relates to the application combinatiilor coordinative in medicine is the use of (m - aqua) - bis (i tricloracetato) - tri (aqua) cobalt aqua cobalt bis (tricloracetato) monohydrate as inhibitor of human myeloid leukaemia.the essence of the invention lies in that as the inhibitor of human myeloid leukaemia's claim (m - aqua) - bis (i tricloracetato) - tri (aqua) cobalt aqua cobalt bis (tricloracetato) monohydrate with formula: the invention consist in determining the (m - aqua) - bis (i tricloracetato) - tri (aqua) cobalt aqua cobalt bis (tricloracetato) monohydrate anticancer activity, which exceeds 1,25...1,35 times characteristics of dimerilor analogues trihidratului aquaetilendiamintetraacetatobismutatului (iii) 1,6 - dinitrotetraamincobalt (iii) and (iii) dihidratului etilendiamintetraacetatobismutatului oxalatotetraamincobalt (iii) (analogue).
机译:本发明涉及组合配合在医学上的应用是(m-水)-双(三氯乙酸)-三(水)钴水合双(三氯乙酸)一水合物作为人骨髓性白血病的抑制剂。本发明的实质在于作为人类髓样白血病的抑制剂要求保护(m-aqua)-双(i tricloracetato)-三(aqua)钴aqua钴双(tricloracetato)一水合物,其分子式为:本发明在于确定(m-aqua)- bis(i tricloracetato)-三(水合钴)钴aqua bis(tricloracetato)一水合抗癌药的活性超过1,25 ... 1,35倍二聚体类似物trihidratului aquaetilendiamintetraacetatobismutatului(iii)的特征1,6--二硝基四氢安那多(iii) (iii)乙二胺二乙胺四乙酸二丁酯草酸四氨基丁酸(iii)(类似物)。

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