首页> 外国专利> N-amp;LCUB; (2S) -4- (3, 4-DIFLUOROBENZYL) MORPHOLIN-2YL!METHYLamp;RCUB; -2-amp;LCUB;3- (METHYLSULPHONYL) AMINO! PHENYLamp;RCUB;ACETAMIDE AS CCR3 ANTAGONIST FOR THE TREATMENT OF INFLAMMATORY CONDITIO

N-amp;LCUB; (2S) -4- (3, 4-DIFLUOROBENZYL) MORPHOLIN-2YL!METHYLamp;RCUB; -2-amp;LCUB;3- (METHYLSULPHONYL) AMINO! PHENYLamp;RCUB;ACETAMIDE AS CCR3 ANTAGONIST FOR THE TREATMENT OF INFLAMMATORY CONDITIO

机译:N-{ (2S)-4-(3,4-二氟联苯)吗啉-2YL! -2-{ 3-(甲基磺酰基)氨基酸!苯乙酰胺为CCR3拮抗剂治疗发炎性症状

摘要

Title: N-{' (2S) -4- (3, 4-DIFLUOROBENZYL) MORPHOLIN-2YL!METHYL} -2-{3-' (METHYLSULPHONYL) AMINO! PHENYL}ACETAMIDE AS CCR3 ANTAGONIST FOR THE TREATMENT OF INFLAMMATORY CONDITIONS[err]Abstract: Compound of formula (I): HsC H H '(0) IIZZ V which is; 3-(f [({[(25)-4-(3,4-dichlorobenzyl)mor-pholin-2-yl]methyl}amino)carbonyl]-amino}methyl)=Nethlylbenzamide; and salts and solvates thereof, a process for its preparation intermediates, pharmaceutical formulations containing it and its use in therapy, as CCR3=antagonist for the treatment of inflammatory conditions.
机译:标题:N- {'(2S)-4-(3,4-二氟联苯)吗啉-2YL!METHYL} -2- {3-'(甲基磺酰基)氨基!苯乙酰胺为CCR3拮抗剂,用于治疗炎症[呃]摘要:式(I)化合物:HsC H H'(0)IIZZ V为: 3-(f [({{((25)-4-(3,4-dichlorophenyl)mor-pholin-2-基]甲基}氨基}羰基]-氨基}甲基)= Nethlylbenzamide;及其盐和溶剂化物,其制备方法制备中间体,包含该中间体的药物制剂及其在治疗中的用途,作为CCR3 =拮抗剂用于治疗炎性疾病。

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