首页> 外国专利> 2-mercapto substituted triazolopyrimidines, methods for preparing them, their use for controlling pathogenic fungi, and medicaments comprising 2-mercapto substituted triazolopyrimidine compounds

2-mercapto substituted triazolopyrimidines, methods for preparing them, their use for controlling pathogenic fungi, and medicaments comprising 2-mercapto substituted triazolopyrimidine compounds

机译:2-巯基取代的三唑并嘧啶,其制备方法,其在控制病原真菌中的用途以及包含2-巯基取代的三唑并嘧啶化合物的药物

摘要

The present invention relates to a process for the preparation of a compound of formula (I) in which the substituents have the following meanings: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkynyloxy A represents hydrogen, hydroxy, alkyl, alkenyl, alkoxy, halogenalkoxy, alkylamino or dialkylamino; m represents 0, 1, 2, 3, 4 or 5; X represents halogen, cyano, alkyl, halogenalkyl, alkoxy or halogenalkoxy; R1And R2Represents a hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkynyl, halogenalkynyl, cycloalkynyl, phenyl or naphthyl, or represents a group of O, N or S A 5-to 10-membered saturated, partially unsaturated or aromatic heterocyclic ring containing 1 to 4 heteroatoms selected from R1And R2Together with the nitrogen atom to which they are attached form a 5-or 6-membered ring wherein the ring is interrupted by an atom selected from the group of O, N and S Alternatively, where R1And / or R2Are optionally substituted as described herein, to 2-mercapto substituted triazolopyrimidines. The invention also relates to a process for preparing the above compound, to a medicament comprising said compound and to their use for controlling phytopathogenic fungi.
机译:本发明涉及一种制备式(I)化合物的方法,其中取代基具有以下含义:L是卤素,氰基,硝基,烷基,烯基,炔基,卤代烷基,卤代烯基,烷氧基,烯氧基,炔氧基A代表氢,羟基,烷基,烯基,烷氧基,卤代烷氧基,烷基氨基或二烷基氨基; m代表0、1、2、3、4或5; X代表卤素,氰基,烷基,卤代烷基,烷氧基或卤素烷氧基; R 1 和R 2 表示氢,烷基,卤代烷基,环烷基,卤代环烷基,烯基,链二烯基,卤素烯基,环烯基,炔基,卤素炔基,环炔基,苯基或萘基,或表示一组O,N或SA的5至10元饱和,部分不饱和或芳族杂环,其中含有1-4个选自R 1 和R 2 一起的杂原子与它们所连接的氮原子形成5元或6元环,其中该环被选自O,N和S的原子中断。或者,其中R 1 And / R 2或R 2 Supre如本文所述任选地被取代为2-巯基取代的三唑并嘧啶。本发明还涉及制备上述化合物的方法,涉及包含所述化合物的药物,以及它们在控制植物病原性真菌中的用途。

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号