首页> 外国专利> New acido 8-ciano-1-cyclopol-7 - (1s, 6s-2, 8-diazabiciclo 4.3.0 nonan-8-il) - 6-fluoro-1, 4-dihydro-4-oxo-3-quinolincarboxilico

New acido 8-ciano-1-cyclopol-7 - (1s, 6s-2, 8-diazabiciclo 4.3.0 nonan-8-il) - 6-fluoro-1, 4-dihydro-4-oxo-3-quinolincarboxilico

机译:新酸8-氰基-1-环酚-7-(1s,6s-2,8-二氮杂双环[4.3.0]壬基-8-基)-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸

摘要

It refers to a very stable pradofloxacino (8-cyano-1-cyclopropene-7 - (1s, 6s-2, 8-diazabiciclo [4.3.0] nonan-8-il) - 6-fluoro-1, 4-dihydro-4-oxo-3-quinolincarboxilic) crystal, which is suitable for Welsh formula. Pradofloxacin, a trihydrate, has an X-ray powder profile with high and medium intensity (more than 30% relative intensity) reflection position (2 theta). Comment more than a month agoAT A TEMPERATURE OF 50 ° OR MORE, A PRADOFLOXACINO SOLUTION IN AN APROTICAL POLAR SOLVENT AND MIX WITH WATER CONTAINING PRADOFLOXACINO TRIHYDRATE SEED CRYSTALS. ALSO REFERRED TO USEFUL PHARMACEUTICAL COMPOSITIONS IN THE TREATMENT OF BACTERIAL DISEASES
机译:它指的是非常稳定的普拉多沙星(8-氰基-1-环丙烯-7-(1s,6s-2,8-二氮杂双[4.3.0]壬基-8-il)-6-氟-1,4-二氢- 4-氧代-3-喹啉羧酸)晶体,适用于威尔士配方。三水合普拉多沙星具有X射线粉末轮廓,具有高和中等强度(相对强度超过30%)的反射位置(2θ)。超过一个月前,在温度为50°C或更高的条件下,在非极性极性溶剂中混合了PRADOFLOXACINO溶液,并用水混合了PRADOFLOXACINO三水合物种子晶体。在细菌性疾病的治疗中还提到了有用的药物成分

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