首页> 外国专利> Pirido - pyrimidine Derivatives, their preparacinn, aplicacinn in Therapeutic

Pirido - pyrimidine Derivatives, their preparacinn, aplicacinn in Therapeutic

机译:Pirido-嘧啶衍生物,其前庭素,阿普卡星在治疗中

摘要

Compounds that respond to the fnrmula (i): in which: - R1 represents an alkyne Group (C1 - C6), a nr2r3 or ch2cor4 Group; R2 and R3 are each independently between, a rtomo of hidrngeno or alkyne (C1 - C6); R4 represents a hydroxyl Group, alkoxy (c1-c4), amino, alquilamino ( C1 - C4)Dialquilamino (c1-c4); r1 represents a radical selected from: - ar2 represents a substituted or non substituted phenyl Group of 1 to 5 times with similar or different substituents selected from a group of rtomo halngeno, alkyl (c1-c4), trifluoromethyl or alkoxy (c1-c4); procedure To preparacinn and aplicacinn in terapcutica.
机译:响应式(i)的化合物:其中:-R1代表炔基(C1-C6),nr2r3或ch2cor4基团; R 2和R 3各自独立地在羟基或炔烃的C 1 -C 6之间。 R4代表羟基,烷氧基(c1-c4),氨基,alquilamino(C1-C4)Dialquilamino(c1-c4); r1代表选自以下的基团:-ar2代表具有类似或不同取代基的1至5倍取代或未取代的苯基,所述取代基选自rt halngeno,烷基(c1-c4),三氟甲基或烷氧基(c1-c4) ;程序在Terapcutica中制备preparacinn和aplicacinn。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号