首页> 外国专利> PYRIDONE-CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND ANTI-TUMOR AGENTS CONTAINING THE PYRIDONE-CARBOXYLIC ACID DERIVATIVES

PYRIDONE-CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND ANTI-TUMOR AGENTS CONTAINING THE PYRIDONE-CARBOXYLIC ACID DERIVATIVES

机译:吡咯烷酮羧酸衍生物,其制备方法和包含吡咯烷酮羧酸衍生物的抗肿瘤剂

摘要

This invention relates to pyridone-carboxylicacid derivatives of the following formula or saltsthereof :whereinR1 is a hydrogen atom, a halogen atom, etc.,R2 is a carboxyl group etc.,R3 is a hydrogen atom etc.,A is a nitrogen atom or CH,m is 1 or 2, aidY is an eliminable group or a group having thefollowing formula:whereinR4 is a hydrogen atom or a lower alkylgroup,Z is a hydrogen atom, a lower alkylgroup, etc.,R5 is a hydrogen atom, a lower alkylgroup, etc.,n is 0 or 1, andp is 1, 2, 3 or 4and to processes for the preparation of these compounds,and further to anti-tumor agents which contain the abovecompounds as effective ingredients.
机译:本发明涉及吡啶酮羧酸下式的酸衍生物或盐其中:其中R 1为氢原子,卤素原子等,R 2为羧基等,R 3为氢原子等,A是氮原子或CHm是1或2,辅助Y是可消除基团或具有公式如下:其中R4是氢原子或低级烷基组,Z是氢原子,低级烷基小组等R5是氢原子,低级烷基小组等n为0或1,并且p是1、2、3或4以及这些化合物的制备方法,以及进一步包含上述成分的抗肿瘤药化合物作为有效成分。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号