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CRYSTALLINE AND AMORPHOUS FORM OF RANOLAZINE AND THE PROCESS FOR MANUFACTURING THEM

机译:纳洛嗪的晶型和非晶态形式及其制备方法

摘要

Process for the preparation of novel crystalline and amorphous form of (±)-1-[3-(2-Methoxyphenoxy)-2-hydroxypropyl]-4-[N-(2,6-dimethylphenyl)carbamoylmethyl] piperazine dihydrochloride & a crystalline form of Ranolazine base is disclosed in the present invention which has the formula (I) and is a medicine useful as anti-anginal agent.
机译:新型(±)-1- [3-(2-甲氧基苯氧基)-2-羟丙基] -4- [N-(2,6-二甲基苯基)氨基甲酰基甲基]哌嗪二盐酸盐的结晶和无定形形式的制备方法及结晶在本发明中公开了具有雷诺嗪碱形式的Ranolazine碱,其具有式(I)并且是用作抗心绞痛药的药物。

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