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Amino Alcohol Derivatives or Phosphonic Acid Derivatives and Pharmaceutical Compositions Containing Indicated Derivatives
Amino Alcohol Derivatives or Phosphonic Acid Derivatives and Pharmaceutical Compositions Containing Indicated Derivatives
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机译:氨基醇衍生物或膦酸衍生物以及含有指示性衍生物的药物组合物
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摘要
An amino alcohol derivative or phosphonic acid derivative each having excellent immunosuppressive activity; a pharmacologically acceptable salt thereof or pharmacologically acceptable ester thereof; and a medicinal composition containing any of these. (I) (In the formula, R1 and R2 each represents hydrogen or an amino-protecting group; R3 represents hydrogen or a hydroxy-protecting group; R4 represents lower alkyl; n is an integer of 1 to 6; X represents oxygen or nitrogen optionally substituted by lower alkyl, etc.; Y represents ethylene; Z represents C1-10 alkylene; R5 represents aryl or substituted aryl; and R6 and R7 each represents hydrogen; provided that when R5 is hydrogen, then Z is neither a single bond nor linear C1-10 alkylene.)
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机译:具有优异的免疫抑制活性的氨基醇衍生物或膦酸衍生物;其药理上可接受的盐或其药理上可接受的酯;以及含有这些成分的药物组合物。 (I)(式中,R 1和R 2分别表示氢或氨基保护基; R 3表示氢或羟基保护基; R 4表示低级烷基; n是1至6的整数; X表示氧或氮Y代表乙烯; Z代表C1-10亚烷基; R5代表芳基或取代的芳基; R6和R7各自代表氢;条件是当R5为氢时,Z既不是单键也不是线性C1-10亚烷基。)
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