Presentation form (obtainable by dissolving indibulin in or with a highly concentrated organic acid), useful to orally administer poorly soluble active compound indibulin, comprises a poorly soluble active compound indibulin

摘要

Presentation form (A) comprises a poorly soluble active compound indibulin (in the form of a supersaturated solution) for oral administration; where (A) is obtainable by dissolving indibulin in or with a highly concentrated organic acid (which is physiologically tolerable per se in diluted form), and diluting by adding water to a physiologically tolerable concentration of the organic acid. Independent claims are also included for: (1) the preparation of (A); and (2) a kit for the simplified handling of the preparation of (A). ACTIVITY : Cytostatic. MECHANISM OF ACTION : Tubulin inhibitor.