首页> 外国专利> CRYSTALLINE FORMS OF 1S-Ä1ALPHA (2S *, 3R *), 9ALPHA-6,10-DIOXO-N- (2-ETHOXY-5-OXO-TETRAHYDRO-3-FURANYL) -9-AE (1-ISOCHINOLYL) CARBONYLENE AMINOÜOCTAHYDRO-6H-PIRIDAZINOÄ1,2-AÜÄ1,2ÜDIAZEPIN-1-carboxamide

CRYSTALLINE FORMS OF 1S-Ä1ALPHA (2S *, 3R *), 9ALPHA-6,10-DIOXO-N- (2-ETHOXY-5-OXO-TETRAHYDRO-3-FURANYL) -9-AE (1-ISOCHINOLYL) CARBONYLENE AMINOÜOCTAHYDRO-6H-PIRIDAZINOÄ1,2-AÜÄ1,2ÜDIAZEPIN-1-carboxamide

机译:1S-Ä1ALPHA(2S *,3R *),9ALPHA-6,10-DIOXO-N-(2-ETHOXY-5-OXO-TETRAHYDRO-3-FURANYL)-9-AE(1-ISOCHINOLYL)羰基氨基甲酸酯-6H-PIRIDAZINOÄ1,2-AÜÄ1,2ÜDIAZEPIN-1-羧酰胺

摘要

Two new crystalline forms of 1S-[1alpha(2S*, 3R*), 9alpha]6, 10-dioxo-N-(2-ethoxy-5-oxo-tetrahydro-3-furany1)-9 [[(1-isoquinolyl) carbony1]amino]octahydro-6H-pyridazino [1,2-a][1,2]diazepin-1-carboxamide (anhydrous or hydrated), their preparation process and the pharmaceutical compositions containing them.
机译:1S- [1α(2S *,3R *),9α6,10-二氧代-N-(2-乙氧基-5-氧代-四氢-3-呋喃基)-9 [[((1-异喹啉基) )羰基[1]氨基]八氢-6H-哒嗪[1,2-a] [1,2]二氮杂-1-甲酰胺(无水或水合),其制备方法和含有它们的药物组合物。

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