首页> 外国专利> Injectable or oral composition comprises azetidine derivatives, polysorbate 80, Solutol HS15 solution and optionally ethanol, propylene glycol or PEG-400 as co-solvent

Injectable or oral composition comprises azetidine derivatives, polysorbate 80, Solutol HS15 solution and optionally ethanol, propylene glycol or PEG-400 as co-solvent

机译:注射剂或口服组合物包含氮杂环丁烷衍生物,聚山梨酸酯80,Solutol HS15溶液和可选的乙醇,丙二醇或PEG-400作为助溶剂

摘要

Injectable or oral composition comprises azetidine derivatives (A), polysorbate 80 (polyethylene glycol monooleate), Solutol HS15 (polyethylene glycol hydroxystearate) and optionally ethanol, propylene glycol or PEG-400 as co-solvent. Injectable or oral composition comprises azetidine derivatives (A) of formula (IA) or (IB), Polysorbate 80 (polyethylene glycol monooleate), Solutol HS15 (polyethylene glycol hydroxystearate) and optionally ethanol, propylene glycol or PEG-400 as co-solvent. Ar = (hetero)aromatic (optionally substituted by 1-4C alkyl, halo, NO, CN, 1-4C alkoxy or OH). [Image].
机译:注射剂或口服组合物包含氮杂环丁烷衍生物(A),聚山梨酸酯80(聚乙二醇单油酸酯),Solutol HS15(聚乙二醇羟基硬脂酸酯)和任选的乙醇,丙二醇或PEG-400作为助溶剂。注射或口服组合物包含式(IA)或(IB)的氮杂环丁烷衍生物(A),聚山梨酯80(聚乙二醇单油酸酯),Solutol HS15(聚乙二醇羟基硬脂酸酯)和任选的乙醇,丙二醇或PEG-400作为助溶剂。 Ar =(杂)芳族(任选地被1-4C烷基,卤素,NO,CN,1-4C烷氧基或OH取代)。 [图片]。

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