首页> 外国专利> A2A Receptor Antagonists and alquinil - 2 - 2 - alquinil pyrazolo - e - 4.3 - 1,2,4 triazolo c - pyrimidine Adenosine 1.5 -

A2A Receptor Antagonists and alquinil - 2 - 2 - alquinil pyrazolo - e - 4.3 - 1,2,4 triazolo c - pyrimidine Adenosine 1.5 -

机译:A2A受体拮抗剂和阿奎尼尔-2-2-阿奎尼尔吡唑并-[e]-4.3-1,2,4三唑并[c]-嘧啶腺苷1.5-

摘要

1. Compounds containing salts of structural formula or drug acceptability shall be independently selected from groups h, hydrocarbyl and ALCOXY in compounds with R of R1, R2, R3, R4 and R5; R6 shall be selected from groups h, hydrocarbyl, hydroxide or ch2f; R7, R8 and R9 shall be selected from groups h respectively, Acoxi, acultio, alcoxidio, alcoxiquie, halo and CF3; Z is R10 arilo, R10 isomerization or R10 is alternative 1-5 selected from independent hydrogen, tar, alquenilo, hidroxi, alcoxi, alcoxi, hydroxi, hydroxil, hidroxil alcoxi, alcoxixy, alcoxi alcoxi acquil groups,1.1.1.1 (DI propoxy) - tar (hydroxy) - methoxyethane, R15 cyclomethoxy, R15 cyclomethylclalquilo, cyclomethoxy oxygen, cyclomethoxy-o-alcoxi, tar-so2 -,Anyone can view this photohalo -CN cianoalquilo -CHF2 -CF3 -OCHF2 -OCF3 -C (O) R13 -O-alquilen-C (O) OR13 -C (O) Oalquilo -N (R11) (R12)N (R11) (R12) -alkyl, N (R11) (R12) -alkoxy, -C (O) N (R13) (R16),Oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen (oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen oxygen -C (= nor17) - tar and - C (= nor17) - CF3; or R10 of two adjacent groups of carbon ring atoms are added together to form - o-ch2-o -,-O- (CH2) 2-O-,...
机译:1.具有R 1,R2,R3,R4和R5的化合物中,具有结构式或药物可接受性盐的化合物应独立选自h,烃基和ALCOXY; R6应选自h,烃基,氢氧化物或ch2f; R7,R8和R9应分别选自h组,Acoxi,acultio,alcoxidio,alcoxiquie,halo和CF3; Z为R10芳基,R10异构化或R10为替代1-5,选自独立的氢,焦油,alquenilo,hidroxi,alcoxi,alcoxi,hydroxi,hydroxil,hidroxil alcoxi,alcoxixy,alcoxi alcoxi acquil基1.1.1.1(DI丙氧基) -焦油(羟基)-甲氧基乙烷,R15环甲氧基,R15环甲基Clalquilo,环甲氧基氧,环甲氧基-邻-alcoxi,tar-so2-,任何人都可以查看此光卤-CN cianoalquilo -CHF2 -CF3 -OCHF2 -OCF3 -C(O)R13 -O-alquilen-C(O)OR13 -C(O)Oalquilo -N(R11)(R12)N(R11)(R12)-烷基,N(R11)(R12)-烷氧基,-C(O)N (R13)(R16),氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气(氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气-氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧气氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧氧-C(= nor17)-焦油和-C(= nor17)-CF3;或两个相邻的碳环原子基团的R10加在一起形成-o-ch2-o-,-O-(CH2)2-O-,...

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