首页> 外国专利> SUBSTITUTED PIPERAZINES (14) DIASZEPINES AND 2,5-DIAZABICYCLO (2,2.1) HEPTANES AS HISTAMINE H1 AND/OR H3 ANTAGONISTS OR HISTAMINE H3 REVERSE ANTAGONISTS

SUBSTITUTED PIPERAZINES (14) DIASZEPINES AND 2,5-DIAZABICYCLO (2,2.1) HEPTANES AS HISTAMINE H1 AND/OR H3 ANTAGONISTS OR HISTAMINE H3 REVERSE ANTAGONISTS

机译:取代的哌嗪(14)地西ZE和2,5-二氮杂双环(2,2.1)庚烷作为组氨酸H1和/或H3拮抗剂或组氨酸H3逆向拮抗剂

摘要

The present invention relates to novel piperazine and azepine derivatives having pharmacological activity, processes for their preparation, to compositions containing them and to their use in the treatment of neurodegenerative disorders including Alzheimer's disease.
机译:本发明涉及具有药理活性的新型哌嗪和氮杂卓衍生物,其制备方法,含有它们的组合物以及它们在治疗神经退行性疾病包括阿尔茨海默氏病中的用途。

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