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METHODS OF INHIBITING PHYSIOLOGICAL CONDITIONS ASSOCIATED WITH AN EXCESS OF NEUROPEPTIDE Y.

机译:抑制与神经肽Y过多有关的生理条件的方法

摘要

A METHOD OF INHIBITING A PHYSIOLOGICAL DISORDER ASSOCIATED WITH AN EXCESS OF NEUROPEPTIDE Y OR ITS SYMPTOMS COMPRISING ADMINISTERING TO A HUMAN IN NEED THEREOF AN EFFECTIVE AMOUNT OF A COMPOUND HAVING THE FORMULA (FORMULA 1)WHEREIN R1 AND R3 ARE INDEPENDENTLY HYDROGEN , O O-CH3, -C-(C1-C6 ALKYL), OR -C-AR, WHEREIN AR IS OPTIONALLY SUBSTITUTED PHENYL;R2 IS SELECTED FROM THE GROUP CONSISTING OF PYRROLIDINE, HEXAMETHYLENEAMINO, AND PIPERIDINO; OR A PHARMACEUTICALLY ACCEPTABLE SALT OF SOLVATE THEREOF.
机译:一种方法,用于抑制与过量人类神经肽Y或其症状有关的,导致人类不适的生理性疾病,从而需要有效量的配方,其中R1和R3中含有R1和R3的配方(式1)。 ,-C-(C1-C6烷基)或-C-AR,其中AR可选地被苯酚取代; R2选自吡咯烷,己二烯基氨基和哌啶子基;或用其制成的药学可接受的盐。

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