FORMULATION OF 6,9-BIS DIMALEATE LIPOSOMES - ((2-AMINOETIL) -AMINO) BENZO (G) ISOQUINOLIN-5,10-DIONA.

摘要

The liposome preparation of the 6,9-bis - [(2- aminoethyl) amino] benzo [g] isoquinolin-5,10-dione dimaleate compound. (BBR 2778) of the formula: characterized in that said liposomes include phosphatidylcholine, cholesterol and the compound BBR 2778 in a weight ratio of cholesterol / phospholipid 1: 2 to 1: 7 and in a weight ratio of BBR 2778 / phospholipid 1: 4 to 1:25.