首页> 外国专利> ((CYCLO)ALKYL SUBSTITUTED)-GAMMA-AMINOBUTYRIC ACID DERIVATIVES (=GABA ANALOGUES), THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS

((CYCLO)ALKYL SUBSTITUTED)-GAMMA-AMINOBUTYRIC ACID DERIVATIVES (=GABA ANALOGUES), THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS

机译:((环)烷基取代的)-γ-氨基丁二酸衍生物(= GABA类似物),其制备及其在治疗神经疾病中的用途

摘要

Novel amines of formulas (1A) and (1B) are disclosed and are useful as agentsin the treatment of epilepsy, faintness attacks,hypokinesia, cranial disorders, neurodegenerative disorders, depression,anxiety, panic, pain, neuropathological disorders, inflammatorydiseases, and gastrointestinal disorders, especially IBS. Processes for thepreparation and intermediates useful in the preparation are alsodisclosed.
机译:公开了式(1A)和(1B)的新型胺,它们可用作试剂在治疗癫痫,昏厥发作,运动障碍,颅骨疾病,神经退行性疾病,抑郁症,焦虑,惊恐,疼痛,神经病理疾病,炎症疾病和胃肠道疾病,尤其是IBS。流程制剂以及可用于该制剂的中间体披露。

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