首页> 外国专利> A PROCESS FOR PREPARATION OF OPTICALLY PURE OR OPTICALLY ENRICHED SULFOXIDE COMPOUNDS, INCLUDING AMORPHOUS ESOMEPRAZOLE AND SALTS THEREOF

A PROCESS FOR PREPARATION OF OPTICALLY PURE OR OPTICALLY ENRICHED SULFOXIDE COMPOUNDS, INCLUDING AMORPHOUS ESOMEPRAZOLE AND SALTS THEREOF

机译:制备光学纯或光学富集的二氧化硫化合物的方法,其中包括无定形的依美拉唑及其盐

摘要

A process of preparation of optically pure or optically enriched isomers of omeprazole and structurally related sulfoxides is provided. Also provided are an amorphous form of esomeprazole, as well a pharmaceutical composition containing it and a method of using it for treatment of gastric disorders.
机译:提供了制备光学纯的或光学富集的奥美拉唑和结构上相关的亚砜的方法。还提供了埃索美拉唑的无定形形式,以及包含其的药物组合物和使用其治疗胃部疾病的方法。

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