首页> 外国专利> Polymorphic forms of (2R, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1h-pyrazol-4-yl) - oxo - 2.6 - dihydro - 1 - (1,2) - 1H indole diazepino (4,5,6 - CD) - 8 (IL - 2R) acetamide, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1h-pyrazol-4-yl) - 2 - oxo - 2.6 - dihydro 1H - 1,2 diazepino 4,5,6 indole - CD - 8 (IL - 2R), (Z) - acetamide 2 - amino - 2 - ciclohex

Polymorphic forms of (2R, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1h-pyrazol-4-yl) - oxo - 2.6 - dihydro - 1 - (1,2) - 1H indole diazepino (4,5,6 - CD) - 8 (IL - 2R) acetamide, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1h-pyrazol-4-yl) - 2 - oxo - 2.6 - dihydro 1H - 1,2 diazepino 4,5,6 indole - CD - 8 (IL - 2R), (Z) - acetamide 2 - amino - 2 - ciclohex

机译:(2R,(Z)-2-氨基-2-环己基-N-(5-(1--甲基-1h-吡唑-4-基)-氧代-2.6-二氢-1-(1,2)的多晶型-1H吲哚重氮(4,5,6-CD)-8(IL-2R)乙酰胺,(Z)-2-氨基-2-环己基-N-(5-(1-甲基-1h-吡唑-4- yl)-2-羰基-2.6-二氢1H-[1,2]二氮杂环庚烷[4,5,6]吲哚-CD-8(IL-2R),(Z)-乙酰胺2-氨基-2-环己基

摘要

Claim 1: a Crystalline form of (2R, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1h-pyrazol-4-yl) - 2 - oxo - 2.6 - dihydro 1H - [1,2] diazepino4,5,6 CD] indole 8 - il) acetamide. Claim 16: an Amorphous form of (2R, (Z) - 2 - amino - 2 - Cyclohexyl - N - (5 - (1 - methyl - 1 - h-pyrazo - 4-yl) - 2 - oxo - 2.6 - dihydro 1H - [1,2] diazepino [4,5,6] indole 8 CD - il) acetamide.Pharmaceutical compositions containing them and their use as Anticancer Therapeutic people.
机译:权利要求1:(2R,(Z)-2-氨基-2-环己基-N-(5-(1-甲基-1h-吡唑-4-基)-2-氧代-2.6-二氢1H- [1,2] diazepino4,5,6 CD]吲哚8-il)乙酰胺。16.非晶态形式的(2R,(Z)-2-氨基-2-环己基-N-(5-(1-甲基) -1-h-吡唑基-4-基)-2-氧代-2.6-二氢1H-[1,2]二氮杂环庚烷[4,5,6]吲哚8 CD-il)乙酰胺。含有它们的药物组合物及其用途抗癌治疗的人。

著录项

  • 公开/公告号AR060348A1

    专利类型

  • 公开/公告日2008-06-11

    原文格式PDF

  • 申请/专利权人 PFIZER PRODUCTS INC.;

    申请/专利号AR2007P101399

  • 发明设计人 RYNBERG RAYMOND;NINKOVIC SACHA;

    申请日2007-04-03

  • 分类号C07D487/06;A61K31/5517;A61K31/407;A61P35/00;C07D487/06;C07D243/00;C07D209/00;

  • 国家 AR

  • 入库时间 2022-08-21 20:08:53

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