首页> 外国专利> agent for the prophylaxis or treatment of metabolic syndrome, method for the prophylaxis or treatment of metabolic syndrome in a mammal, and use of 2-ethoxy-1- 2 '- (5-oxo-2,5-dihydro- 1,2,4-oxadiazol-3-yl) biphenyl-4-yl methyl -1h-benzimidazol-7-carboxylic acid or a salt thereof or a prodrug thereof in combination with a ppargam agonist-like substance

agent for the prophylaxis or treatment of metabolic syndrome, method for the prophylaxis or treatment of metabolic syndrome in a mammal, and use of 2-ethoxy-1- 2 '- (5-oxo-2,5-dihydro- 1,2,4-oxadiazol-3-yl) biphenyl-4-yl methyl -1h-benzimidazol-7-carboxylic acid or a salt thereof or a prodrug thereof in combination with a ppargam agonist-like substance

机译:预防或治疗代谢综合症的药物,预防或治疗哺乳动物代谢综合症的方法,以及2-乙氧基-1- [[2'-((5-oxo-2,5-dihydro-1, 2,4-恶二唑-3-基)联苯基-4-基]甲基] -1h-苯并咪唑-7-羧酸或其盐或前药与苯丙胺激动剂样物质组合

摘要

AGENT FOR PROPHYLAXY OR TREATMENT OF METABOLIC SYNDROME, METHOD FOR PROPHYLAXY OR TREATMENT OF METABOLIC SYNDROME IN A MAMMAL, AND, USE OF 2-ETHIOXY-1- ¢ -2 '- (5-OXY-2,5-DIID) 1,2,4-OXADIAZOL-3-IL) BIFENI L-4-IL! METHYL -1H-BENZIMIDAZOL-7-CARBOXYLIC OR A SALT OF THE SAME OR A PRODUCT OF THE SAME IN COMBINATION WITH A SUBSTANCE SIMILAR TO THE AGONIST PPARGAMA. The present invention provides an agent for the prophylaxis or treatment of metabolic syndrome comprising (2-ethoxy-1- ¢ an 2 '- (5-oxo-2,5-dihydro-1,2,4-oxadiazole-3-acid). il) biphenyl-4-ylmethyl-1 H -benzimidazol-7 carboxylic acid or a salt thereof or a prodrug thereof and a PPAR agonist-like substance in combination.
机译:代谢综合征的预防或治疗代理商,哺乳动物代谢综合征的预防或治疗方法,以及使用2-ETHIOXY-1-¢-2'-(5-OXY-2,5-DIID)1,2 ,4-OXADIAZOL-3-IL)BIFENI L-4-IL!甲基-1H-苯并咪唑-7-羧酸或其盐或该产品的盐,与类似抗精神病药的物质结合使用。本发明提供了一种预防或治疗代谢综合征的药物,其包含(2-乙氧基-1-¢2'-(5-氧代-2,5-二氢-1,2,4-氧二唑-3-酸) il)联苯基-4-基甲基-1H-苯并咪唑-7羧酸或其盐或其前药与PPAR激动剂样物质组合。

著录项

  • 公开/公告号BRPI0516246A

    专利类型

  • 公开/公告日2008-08-26

    原文格式PDF

  • 申请/专利权人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;

    申请/专利号BR2005PI16246

  • 发明设计人 NOBUHIRO NISHIGAKI;

    申请日2005-10-06

  • 分类号A61K31/19;

  • 国家 BR

  • 入库时间 2022-08-21 20:08:44

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