首页>
外国专利>
CONJUGATES COMPRISING AN ANTITUMOUR AGENT AND THEIR USE
CONJUGATES COMPRISING AN ANTITUMOUR AGENT AND THEIR USE
展开▼
机译:组成一个反倾销代理人及其使用
展开▼
页面导航
摘要
著录项
相似文献
摘要
Prodrugs of formula W-Z-M (I) are new:. M = label or therapeutic agent having an active intracellular site (SA); W-Z is a ligand, comprising arm Z and end gp. W; the bond between Z and M inhibits intracellular penetration of (I) and/or inhibits expression of marker-M, and this bond is cleaved selectively by factors secreted by target cells such that M can then be expressed or can enter the cell; W ensures stability of (I) in serum and circulating blood.
展开▼
机译:式W-Z-M(I)的前药是新的:。 M =具有活性细胞内位点(SA)的标记或治疗剂; W-Z是配体,包括臂Z和末端gp。 W; Z和M之间的键抑制(I)的细胞内渗透和/或抑制标记物M的表达,并且该键被靶细胞分泌的因子选择性地切割,从而M可以表达或可以进入细胞。 W确保(I)在血清和循环血液中的稳定性。
展开▼