首页> 外国专利> SUBSTITUTED ISOQUINOLINE-1,3(2H,4H)-DIONES, 1-THIOXO-1,4-DIHYDRO-2H-ISOQUINOLINE-3-ONES AND 1,4-DIHYDRO-3(2H)-ISOQUINOLONES AND USE THEREOF AS KINASE INHIBITOR

SUBSTITUTED ISOQUINOLINE-1,3(2H,4H)-DIONES, 1-THIOXO-1,4-DIHYDRO-2H-ISOQUINOLINE-3-ONES AND 1,4-DIHYDRO-3(2H)-ISOQUINOLONES AND USE THEREOF AS KINASE INHIBITOR

机译:取代的异喹啉-1,3(2H,4H)-二酮,1-硫代-1,4-二氢-2H-异喹啉-3-酮和1,4-二氢-3(2H)-异戊二酮并将其用作激酶抑制剂

摘要

This invention provides compounds of Formula (I), having the structure where GSUP1/SUP, GSUP2/SUP, GSUP3/SUP, GSUP4/SUP, ASUP1/SUP, ASUP2/SUP, YSUP1/SUP, YSUP2/SUP, LSUP1/SUP, Z, e and f are defined herein, or a pharmaceutically acceptable salt thereof, which are useful for treating or preventing cancer.
机译:本发明提供了具有结构式(I)的化合物,其中G 1 ,G 2 ,G 3 ,G 4 < / SUP>,A 1 ,A 2 ,Y 1 ,Y 2 ,L 1 <本文定义了/ ZUP,Z,e和f,或其药学上可接受的盐,其可用于治疗或预防癌症。

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