首页> 外国专利> USE OF KYNURENIC ACID AND DERIVATIVES THEREOF IN THE TREATMENT OF CONDITIONS OF THE GASTROINTESTINAL TRACT ACCOMPANIED BY HYPERMOTILITY AND INFLAMMATION OR GOUT OR MULTIPLE SCLEROSIS

USE OF KYNURENIC ACID AND DERIVATIVES THEREOF IN THE TREATMENT OF CONDITIONS OF THE GASTROINTESTINAL TRACT ACCOMPANIED BY HYPERMOTILITY AND INFLAMMATION OR GOUT OR MULTIPLE SCLEROSIS

机译:动酸及其衍生物在治疗胃功能不全和发炎或痛风或多发性菌血症伴发的胃肠道疾病中的应用

摘要

The subject of the invention is the use of kynurenic acid (KYNA) and its derivatives and physiologically acceptable salts of the general formula (I) in the manufacture of a medicament for the treatment of conditions characterized by pathophysiological conditions of the GI tract accompanied by increased motility and an elevated activity of the enzyme xanthine oxidoreductase (XOR), and further for the treatment of gout or multiple sclerosis. The meanings of the substituents of general formula (I) are defined in the claims.
机译:本发明的主题是犬尿酸(KYNA)及其衍生物和通式(I)的生理上可接受的盐在制备药物中的用途,所述药物用于治疗以胃肠道的病理生理学状况为特征并伴有病情恶化的疾病。黄嘌呤氧化还原酶(XOR)的运动性和较高的活性,进一步用于治疗痛风或多发性硬化症。通式(I)的取代基的含义在权利要求中定义。

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