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PHARMACEUTICAL FORMULATIONS COMPRISING A LONG-ACTING BETA2-AGONIST FOR ADMINISTRATION BY NEBULISATION

机译:包含长效β2-激动剂的药理配方,可通过雾化进行管理

摘要

The invention relates to a liquid, propellant-free pharmaceutical formulation in the form of ready-to-use preparation for administration by nebulisation comprising a water soluble salt of the betaSUB2/SUB-agonist 8-hydroxy-5-[1-hydroxy-2-[[2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]-2(1H)-quinolinone as active ingredient. The active ingredient is chemically stable in the formulation, and said formulation is provided of an adequate shelf-life suitable for commercial distribution, storage and use.
机译:本发明涉及一种液体形式的,无推进剂的药物制剂,该制剂以喷雾形式给药,其包含β 2 激动剂8-羟基-5-5的水溶性盐。作为活性成分的[1-羟基-2-[[[2-(4-甲氧基苯基)-1-甲基乙基]氨基]乙基] -2(1H)-喹啉酮。活性成分在制剂中是化学稳定的,并且所述制剂具有适合于商业分配,储存和使用的足够的保存期限。

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