首页> 外国专利> COMPOUNDS CONTAINING N-HETEROARYRYL RESIDUE ASSOCIATED WITH CONDENSED CYCLIC RESIDUES FOR INHIBITION OF NAD (P) H-OXIDASES AND ACTIVATION OF PLATELETS

COMPOUNDS CONTAINING N-HETEROARYRYL RESIDUE ASSOCIATED WITH CONDENSED CYCLIC RESIDUES FOR INHIBITION OF NAD (P) H-OXIDASES AND ACTIVATION OF PLATELETS

机译:包含N-杂芳基残基与稠合循环残基相关的化合物,可抑制NAD(P)H-氧化酶和激活血小板

摘要

The invention relates to compounds containing a N-heteroaryl moiety, which is linked via oxygen, sulfur or nitrogen, or via a methylene bridge and oxygen, sulfur or nitrogen to a fused ring moiety, in particular to the 1,2,3-triazoloÄ4,5-dÜpyrimidine-7-yl radical. The invention also relates to a process for the preparation of said compounds and the use thereof in drugs for the treatment of NAD(P)H oxidases-related diseases and disorders and inhibition of platelet activation.
机译:本发明涉及含有N-杂芳基部分的化合物,该部分通过氧,硫或氮或通过亚甲基桥与氧,硫或氮连接到稠合的环部分上,特别是1,2,3-三唑并4 ,5-5-嘧啶-7-基团。本发明还涉及所述化合物的制备方法及其在治疗NAD(P)H氧化酶相关疾病和病症以及抑制血小板活化的药物中的用途。

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