首页> 外国专利> SELECTIVE NPY (Y5) ANTAGONISTS

SELECTIVE NPY (Y5) ANTAGONISTS

机译:选择性NPY(Y5)拮抗剂

摘要

This invention is directed to triazine derivatives, bicyclic compounds and tricyclic compounds which are selective antagonists for a NPY (Y5) receptor. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of a compound of the invention and a pharmaceutically acceptable carrier. This invention provides a pharmaceutical composition made by combining a therapeutically effective amount of a compound of this invention and a pharmaceutically acceptable carrier. This invention provides a process for making a pharmaceutical composition comprising combining a therapeutically effective amount of a compound of the invention and a pharmaceutically acceptable carrier. The invention further provides the use of a compound of the invention for the preparation of a pharmaceutical composition for treating an abnormality, wherein the abnormality is alleviated by decreasing the activity of a human Y5 receptor.
机译:本发明涉及三嗪衍生物,双环化合物和三环化合物,它们是NPY(Y5)受体的选择性拮抗剂。本发明提供了药物组合物,其包含治疗有效量的本发明的化合物和药学上可接受的载体。本发明提供了通过将治疗有效量的本发明化合物与药学上可接受的载体结合而制成的药物组合物。本发明提供了制备药物组合物的方法,该方法包括将治疗有效量的本发明化合物与药学上可接受的载体混合。本发明进一步提供本发明的化合物在制备用于治疗异常的药物组合物中的用途,其中所述异常通过降低人Y5受体的活性而减轻。

著录项

  • 公开/公告号DE60034783T2

    专利类型

  • 公开/公告日2008-01-31

    原文格式PDF

  • 申请/专利权人 H. LUNDBECK A/S VALBY;

    申请/专利号DE2000634783T

  • 发明设计人

    申请日2000-04-21

  • 分类号C07D251/70;C07D403/12;C07D401/12;C07D413/12;C07D409/12;C07D417/12;C07D403/04;C07D251/50;C07D251/44;A61K31/53;A61P3/04;

  • 国家 DE

  • 入库时间 2022-08-21 19:48:34

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号