首页> 外国专利> NOVEL PIPERAZINE AND PIPERIDINE DERIVATIVES AS INHIBITORS OF TYPE 3 17BETA-HYDROXYSTEROID DEHYDROGENASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME FOR THE TREATMENT OF ANDROGEN DEPENDENT DISEASES

NOVEL PIPERAZINE AND PIPERIDINE DERIVATIVES AS INHIBITORS OF TYPE 3 17BETA-HYDROXYSTEROID DEHYDROGENASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME FOR THE TREATMENT OF ANDROGEN DEPENDENT DISEASES

机译:新型哌嗪和哌啶衍生物作为3型17-羟基-羟甾体脱氢酶和药物组合物的抑制剂,可治疗雄激素相关疾病

摘要

There are disclosed compounds of the formula (I): prodrugs thereof, or pharmaceutically acceptable salts of the compounds or of said prodrugs which are useful as inhibitors of Type 3 17beta-Hydroxysteroid Dehydrogenase. Also disclosed are pharmaceutical compositions containing said compounds and their use for the treatment or prevention of androgen dependent diseases.
机译:公开了式(I)的化合物:其前药,或该化合物或所述前药的药学上可接受的盐,其可用作3型17β-羟基类固醇脱氢酶的抑制剂。还公开了包含所述化合物的药物组合物及其在治疗或预防雄激素依赖性疾病中的用途。

著录项

  • 公开/公告号IL160065B

    专利类型

  • 公开/公告日2009-07-20

    原文格式PDF

  • 申请/专利权人 SCHERING CORPORATION;

    申请/专利号IL160065

  • 发明设计人

    申请日2004-01-26

  • 分类号C07D211/22;A61K31/445;A61K31/496;A61P5/26;A61P13/08;A61P15/08;A61P17/00;A61P17/10;A61P17/14;A61P35/00;A61P43/00;C07D211/34;C07D211/48;C07D295/185;C07D401/06;C07D401/12;C07D401/14;C07D405/12;C07D409/02;C07D409/12;C07D409/14;C07D417/12;C07D417/14;

  • 国家 IL

  • 入库时间 2022-08-21 19:27:47

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