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PROCESS FOR THE PREPARATION OF AN ANTIBACTERIAL QUINOLONE COMPOUND

机译:抗菌喹诺酮类化合物的制备方法

摘要

It comprises a process for the preparation of levofloxacin based on a cyclisation reaction of a compound of formula (IV), which has the alcohol group protected, followed by a deprotection reaction and the conversion of the compound obtained to levofloxacin by a process comprising a hydrolysis reaction and a second cyclisation reaction. It also comprises new intermediates compounds.;
机译:它包括基于具有被保护的醇基的式(IV)化合物的环化反应制备左氧氟沙星的方法,然后进行脱保护反应,并通过包含水解的方法将所得化合物转化为左氧氟沙星反应和第二个环化反应。它还包括新的中间体化合物。

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