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Oxazolidinone Compounds, its polymorphic forms, processes for preparing such polymorphic forms, Pharmaceutical compositions containing them and Uses Thereof for the treatment of bacterial infections
Oxazolidinone Compounds, its polymorphic forms, processes for preparing such polymorphic forms, Pharmaceutical compositions containing them and Uses Thereof for the treatment of bacterial infections
This provides a compound of formula (1), in Crystalline form, or any of its enantiomers or mixtures thereof, or pharmaceutically acceptable salts or solvates, for use as a Drug, The Compound of formula (1) is active against human pathogens and Gram - Veterinary Some Gram - positive and negative with a weak Inhibitory activity of monoamine oxidase (MAO).They are useful for the treatment of bacterial infections. This also describes forms of the compound (S) - N - [3 - [4 - (Cyano piperidin - 1 - 3 - fluoro - II) phenyl] - 2 - oxo - 5 - methyl - oxazolidin} acetamide.Claim 1: a compound of formula (1), or any of its enantiomers or mixtures thereof, or pharmaceutically acceptable salts or solvates, characterized in that it is used as a Medicine.Claim 3: a polymorphic form, called a form B of a compound according to claim 1, characterized in that it comprises an x-ray diffractogram Peaks approximately 13.4 6.4; characteristic; and 24.6 degrees two Theta.Claim 1: a polymorphic form, called a compound form, according to claim 1, characterized in that it comprises an x-ray diffractogram Peaks characteristic of Greater Intensity than the rest to approximately 16.6 7.1; and 23.2 degrees two Theta.Claim 1: a polymorphic Form C, called a compound form, according to claim 1, characterized in that it comprises an x-ray diffractogram Peaks approximately 8.8 9.5; characteristic; 14.4; 20.3 23.0 degrees; and 2 Theta.
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