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COVALENTLY BRIDGED INSULIN DIMERS

机译:共价桥接的胰岛素稀释剂

摘要

The invention relates to insulin analogues of formula (I), in which X canindependently be a branched or unbranchedC1-C10-alkyl group, a simply or multiply substituted aryl group, a C1-C10-alkyl group, simply or multiply substituted or unsubstitutedO-aryl group, an amino acid or a derivative thereof, or a group of the formulaNRR'; R, R' is H, NH2, a branched or unbranchedC1-C10-alkyl rest or a simply or multiply substituted or unsubstituted arylgroup; and n is 0, 1, 2,... 16. The invention also relates toa medicament containing such insulin analogues, a method for preparing amedicament for the treatment of diabetes and a methodfor the preparation of insulin analogues.
机译:本发明涉及式(I)的胰岛素类似物,其中X可以独立地是分支机构或不分支机构C1-C10-烷基,简单或多取代的芳基,C1-C10-烷基,简单或多取代或未取代O-芳基,氨基酸或其衍生物或下式的基团NRR'; R,R'为H,NH2,支链或直链C 1 -C 10烷基残基或简单或多取代或未取代的芳基组;并且n是0、1、2,... 16。本发明还涉及含有此类胰岛素类似物的药物,用于治疗糖尿病的药物和方法用于制备胰岛素类似物。

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