首页> 外国专利> 6, 7 -DIHYDRO- 5H- PYRROLO 3, 4-D PYRIMIDIN-4-YL -QUINOLIN-3 -YLAMINE COMPOUNDS USEFUL AS FAAH MODULATORS AND USES THEREOF

6, 7 -DIHYDRO- 5H- PYRROLO 3, 4-D PYRIMIDIN-4-YL -QUINOLIN-3 -YLAMINE COMPOUNDS USEFUL AS FAAH MODULATORS AND USES THEREOF

机译:6,7-二氢-5H-吡咯[3,4-D]吡喃酮-4-基]-喹诺林-3-基胺化合物,可用作FAAH调节剂并使用它们

摘要

Compounds are disclosed that have formula I: where A, B, L1, W, Y, R1, and R3are as defined herein. The com-pounds and pharmaceutical compositions thereof are useful for the preventionand treatment of a variety of conditions in mammalsincluding humans, including by way of non- limiting example, pain, anxiety,depression, inflammation, cognitive disorders,weight and eating disorders, Parkinson's disease, Alzheimer's disease,spasticity, addiction, glaucoma, and others.
机译:公开了具有式I的化合物:其中A,B,L1,W,Y,R1和R3如本文所定义。 com-磅及其药物组合物可用于预防和治疗哺乳动物的各种疾病包括人类,包括但不限于疼痛,焦虑,抑郁症,炎症,认知障碍,体重和饮食失调,帕金森氏病,阿尔茨海默氏病,痉挛,成瘾,青光眼等。

著录项

  • 公开/公告号CA2744343A1

    专利类型

  • 公开/公告日2010-05-27

    原文格式PDF

  • 申请/专利权人 RENOVIS INC.;

    申请/专利号CA20092744343

  • 申请日2009-11-17

  • 分类号C07D487/04;A61K31/519;A61P9;A61P11;A61P19/02;A61P25;

  • 国家 CA

  • 入库时间 2022-08-21 18:42:12

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