首页> 外国专利> 2-{-3-2-(PHENYL)-OXAZOL-4-YLMETHOXYMETHYL!-CYCLOHEXYLMETHOXY };-PROPIONIC ACID DERIVATIVES USED AS PPAR LIGANDES (PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS) FOR THE TREATMENT OF HYPERLIPIDAEMIE AND DIABETES

2-{-3-2-(PHENYL)-OXAZOL-4-YLMETHOXYMETHYL!-CYCLOHEXYLMETHOXY };-PROPIONIC ACID DERIVATIVES USED AS PPAR LIGANDES (PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS) FOR THE TREATMENT OF HYPERLIPIDAEMIE AND DIABETES

机译:2-{-3-2-(Phenyl)-oxazol-4-ylmethoxoxymethethyl!-cyhexhexylmethhooxy};-用作PPAR配体的丙酸衍生物(过氧肟酸增生剂活化的受体)用于治疗高脂血症和糖尿病

摘要

The present invention comprises compounds and compositions for the treatment of metabolic disorders and more particularly, those insulin-related metabolic disorders of the blood such as hyperlipidemia, diabetes, insulin-resistance and the like comprising acetic acid derivatives with cyclohexylmethoxy substituents and their salts. Known as peroxisome proliferator-activated receptors (PPAR) agonists/antagonists, the invention relates to compounds of the formula I wherein the various substituent R-groups are more specifically defined herein.
机译:本发明包括用于治疗代谢紊乱的化合物和组合物,更具体地讲,包括与具有环己基甲氧基取代基的乙酸衍生物和其盐有关的那些与胰岛素相关的血液代谢紊乱,例如高脂血症,糖尿病,胰岛素抵抗等。被称为过氧化物酶体增殖物激活的受体(PPAR)激动剂/拮抗剂,本发明涉及式I的化合物,其中各种取代基R-基团在本文中更具体地定义。

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