首页> 外国专利> Use of compound acid (+) 1,4 - dihydro - 7 - (3S, 4S) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolid inil - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carboxu00eclico enantiomericamente pure, and compound acid (+) 1,4 - dihydro - 7 - (3S, 4S) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolidi nil - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carbo Xu00eclico enantiomericamente pure

Use of compound acid (+) 1,4 - dihydro - 7 - (3S, 4S) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolid inil - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carboxu00eclico enantiomericamente pure, and compound acid (+) 1,4 - dihydro - 7 - (3S, 4S) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolidi nil - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carbo Xu00eclico enantiomericamente pure

机译:使用化合物酸(+)1,4-二氢-7-[(3S,4S)-3-甲基-4-(甲基氨基)-1吡咯烷酮]-4-氧代-1-(2-( 2-氨基-4-噻唑基)-1,8-naftiridina-3-羧基对映体纯和复合酸(+)1,4-二氢-7-(3S,4S)-3-甲基-4 -(甲基氨基)-1-吡咯烷无]-4-氧代-1-(2-(2-氨基-4-噻唑基)-1,8-萘啶酮-3-碳X u00eclico对映异构纯

摘要

Use of compound acid (+) 1,4 - dihydro - 7 - [(3S, 4S) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolid inil] - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carboxilico enantiomericamente pure, and compound acid (+) 1,4 - dihydro - 7 - (3S, 4S) - 3 - methoxy - 4 - (methylamino) - 1 - pirrolidinil] - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina carbox - 3 - u00eclico enantiomericamente pure "methods of treatment, prevention or control of cancer,Including some leukemias, are described. The methods comprise the administration of acid (+) 1, 4 - dihydro - 7 - (3S, 4 (s) - 3 - metu00f3xi - 4 - (methylamino) - 1 - pirrolidinil] - 4 - oxo - 1 - (2 - (2-amino-4-thiazolyl) - 1,8 - naftiridina - 3 - carboxylic enantiomericamente pure. Methods are also provided with detection using this compound with chemotherapy, radiation therapy, hormonal therapy, biological therapy or immunotherapy.Pharmaceutical compositions and single unit dosage forms suitable for use in such methods are also described.
机译:使用化合物酸(+)1,4-二氢-7-[(3S,4S)-3-甲基-4-(甲基氨基)-1吡咯烷酮]-4-氧代-1-(2-( 2-氨基-4-噻唑基)-1,8-naftiridina-3-羧基对映体纯和复合酸(+)1,4-二氢-7-(3S,4S)-3-甲氧基-4-(甲氨基) -1-吡咯烷腈]-4-氧代-1-(2-(2-氨基-4-噻唑基)-1,8-naftiridina羧化物-3-纯的“对映体”治疗,预防或控制癌症的方法,描述了包括一些白血病的方法,该方法包括施用酸(+)1,4-二氢-7-(3S,4(s)-3-met u00f3xi-4-(甲氨基)-1-吡咯烷腈]- 4-氧代-1-(2-(2-氨基-4-噻唑基)-1,8-萘啶酮-3-羧基对映体纯。使用该化合物的检测方法也包括化学疗法,放射疗法,激素疗法,生物学治疗或免疫治疗药物组合物和适合的单单位剂型或在这种方法中的使用也进行了描述。

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