首页> 外国专利> USE OF ESTERS OF L-CARNITINE OR ALKANOYL L-CARNITINES FOR THE PREPARATION OF A LIPOSOME FOR THE TRANSPORT OF A NATURALLY OCCURING OR MODIFIED PLASMID OR POLYNUCLEOTIDE AND COMPOSITIONS COMPRISING THE SAME

USE OF ESTERS OF L-CARNITINE OR ALKANOYL L-CARNITINES FOR THE PREPARATION OF A LIPOSOME FOR THE TRANSPORT OF A NATURALLY OCCURING OR MODIFIED PLASMID OR POLYNUCLEOTIDE AND COMPOSITIONS COMPRISING THE SAME

机译:左旋肉碱或烷基左旋肉碱的酯在制备脂质体中的用途,所述脂质体用于运输天然或修饰的质粒或多聚核苷酸及其组成

摘要

The use of esters of L-carnitine and alkanoyl L-carnitines as cationic lipids for the intracellular delivery of pharmacologically active compounds is described. The esters according to the invention have general formula (II) CHEM wherein the R groups are as defined in the description.
机译:描述了L-肉碱和烷酰基L-肉碱的酯作为阳离子脂质用于药理活性化合物的细胞内递送的用途。根据本发明的酯具有通式(II),其中R基团如说明书中所定义。

著录项

  • 公开/公告号IL175366A

    专利类型

  • 公开/公告日2010-12-30

    原文格式PDF

  • 申请/专利号IL20060175366

  • 发明设计人

    申请日2006-05-01

  • 分类号C07C229;A61K8;A61K8/11;A61K8/14;A61K8/30;A61K8/37;A61K8/44;A61K9/127;A61K31/225;A61K31/337;A61K31/4745;A61K39;A61K45;A61K47/18;A61K47/24;A61K47/44;A61K48;A61P35;A61Q19;C07C229/02;C07C229/22;

  • 国家 IL

  • 入库时间 2022-08-21 18:06:25

相似文献

  • 专利
  • 外文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号