首页> 外国专利> AMINO SUBTITIUTED BENZOYL DERIVATIVES, METHODS FOR THEIR PREPARATION AND THEIR USE IN THE PREPARATION OF ANTI-VIRUS DRUGS

AMINO SUBTITIUTED BENZOYL DERIVATIVES, METHODS FOR THEIR PREPARATION AND THEIR USE IN THE PREPARATION OF ANTI-VIRUS DRUGS

机译:氨基取代的苯甲酰衍生物,其制备方法及其在制备抗病毒药物中的用途

摘要

A group of amino substituted benzoyl derivatives, their preparation and their use. The screening and research on an antiviral drug with hA3G/Vif as a target point proves that the 3-amino benzoyl derivatives not only have the combined activity for the hA3G/Vif, but also have a function of inhibiting replication of viruses. The present invention provides the possible breakthrough progress for the problem of HIV drug resistance, thereby providing a novel clinical antiviral drug which has higher efficiency.
机译:一组氨基取代的苯甲酰基衍生物,其制备和用途。以hA3G / Vif为靶点的抗病毒药物的筛选和研究证明,3-氨基苯甲酰基衍生物不仅具有对hA3G / Vif的联合活性,而且具有抑制病毒复制的功能。本发明为HIV耐药性问题提供了可能的突破性进展,从而提供了一种效率更高的新型临床抗病毒药物。

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