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COMPOSITION OF MOLECULAR ELEMENTS FOR PHOSPHORYLASE KINASE INHIBITION

机译:磷酸激酶激酶抑制分子元素的组成

摘要

Symmetrical curcuminoids molecular compounds that have been found to have anti-injury activity. It has been shown to benefit burns and photodamaged skin. The improvement is mediated via inhibition of phosphorylase kinase activity. Phosphorylase kinase is released within 3 minutes following injury. Blocking the elevated phosphorylase kinase activity released after injury by phosphorylase kinase inhibitiors, such as symmetrical curcuminoids, results in rapid reversal of burns injury and repair of photodamaged skin.
机译:已发现对称的姜黄素分子化合物具有抗损伤活性。已证明它有益于烧伤和光损伤的皮肤。该改善是通过抑制磷酸化酶激酶活性来介导的。磷酸酶激酶在受伤后3分钟内释放。阻断损伤后由对称的姜黄素等磷酸化酶激酶抑制剂释放的升高的磷酸化酶激酶活性,导致烧伤迅速逆转并修复光损伤的皮肤。

著录项

  • 公开/公告号WO2011084129A1

    专利类型

  • 公开/公告日2011-07-14

    原文格式PDF

  • 申请/专利权人 HENG MADALENE C.Y.;

    申请/专利号WO2010US03135

  • 发明设计人 HENG MADALENE C.Y.;

    申请日2010-12-08

  • 分类号A01N35;

  • 国家 WO

  • 入库时间 2022-08-21 17:56:43

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